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benzimidazoles veterinarios

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benzimidazoles veterinarios

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benzimidazoles veterinarios farmacologia 2

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benzimidazoles veterinariosOnline version

benzimidazoles veterinarios farmacologia 2

by Nathalie Sadjey Davila Roa
1

Los benzimidazoles actúan uniéndose a la ? - del parásito , impidiendo la formación de y causando alteraciones en el transporte de .

2

El y el son benzimidazoles usados en medicina veterinaria para el control de nematodos .

3

La resistencia a benzimidazoles en nematodos gastrointestinales se asocia principalmente con ? - , especialmente en los codones , y , lo que disminuye la afinidad del fármaco .

4

Un ejemplo de benzimidazol utilizado en rumiantes es el y el

5

El albendazol está contraindicado durante la debido a efectos teratogénicos .

6

La muerte del parásito ocurre por energético debido a la falta de

7

Tras su administración oral , muchos benzimidazoles presentan , alta y requieren para generar metabolitos activos .

8

El albendazol se metaboliza a , considerado el principal , responsable de su eficacia contra parásitos tisulares .

9

En rumiantes , la eficacia terapéutica de los benzimidazoles puede aumentar debido al , lo que favorece una .

10

Los benzimidazoles ejercen su acción antihelmíntica mediante la unión selectiva a la ? - , inhibiendo la , lo que provoca alteración en el transporte intracelular de , disminución en la absorción de , agotamiento progresivo de las reservas de , reducción en la síntesis de y finalmente degeneración estructural del , conduciendo a su inmovilización y eliminación por el hospedador .

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